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Zacopride hydrochloride

CAS No. 101303-98-4

Zacopride hydrochloride ( —— )

Catalog No. M20083 CAS No. 101303-98-4

Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 132 In Stock
25MG 267 In Stock
50MG 430 In Stock
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Biological Information

  • Product Name
    Zacopride hydrochloride
  • Note
    Research use only not for human use.
  • Brief Description
    Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
  • Description
    Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT3 antagonist; 5-HT4 agonist; IK1/Kir2.1 agonist
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    101303-98-4
  • Formula Weight
    346.26
  • Molecular Formula
    C15H20ClN3O2.HCl
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    Cl.COc1cc(N)c(Cl)cc1C(=O)NC1CN2CCC1CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Nagakura Y et al. Pharmacological properties of a novel gastrointestinal prokinetic benzamide selective for human 5-HT4 receptor versus human 5-HT3 receptor. Pharmacol Res. 1999 May;39(5):375-82.
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